Tuning reactivity of glycosyl imidinium intermediate for 2-azido-2-deoxyglycosyl donors in α-glycosidic bond formation

Arun B. Ingle, Chin Sheng Chao, Wei Cheng Hung, Kwok-Kong Mong*

*Corresponding author for this work

Research output: Contribution to journalArticlepeer-review

34 Scopus citations

Abstract

The chemical properties of nucleophile additives were investigated in a modulated glycosylation context. N-Formylmorpholine (NFM) was found to be an effective modulator for glycosylation with less reactive 2-azido-2- deoxythioglucosyl and thiogalactosyl donors.

Original languageEnglish
Pages (from-to)5290-5293
Number of pages4
JournalOrganic Letters
Volume15
Issue number20
DOIs
StatePublished - 18 Oct 2013

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